- 847950-09-8
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Structure-based design of novel 2-amino-6-phenyl-pyrimido[5′, 4′:5,6]pyrimido[1,2-a]benzimidazol-5(6H)-ones as potent and orally active inhibitors of lymphocyte specific kinase (Lck): Synthesis, SAR, and in vivo anti-inflammatory activity
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Journal of Medicinal Chemistry p. 1637 - 1648
(2008/12/22)
- File number:2
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- 847952-36-7
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Design, synthesis, and structure-activity relationship study of bicyclic piperazine analogs of indole-3-carboxamides as novel cannabinoid CB1 receptor agonists
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Bioorganic and Medicinal Chemistry Letters p. 7327 - 7330
(2011/01/12)
- File number:6
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- 847974-76-9
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Alkylation of Nitropyridines via Vicarious Nucleophilic Substitution
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Organic Letters p. 516 - 519
(2022/01/20)
- File number:2
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- 84799-98-4
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Chiral oxazoline-1,3-dithianes: New effective nitrogen-sulfur donating ligands in asymmetric catalysis
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Tetrahedron Asymmetry p. 3232 - 3240
(2007/10/03)
- File number:4
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- 84800-62-4
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Tuned-affinity bivalent ligands for the characterization of opioid receptor heteromers
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ACS Medicinal Chemistry Letters p. 640 - 644,5
(2020/08/31)
- File number:6
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- 848029-08-3
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Solid supported synthesis of structurally diverse dihydropyrido[2,3-d] pyrimidines using microwave irradiation
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Tetrahedron Letters p. 1345 - 1348
(2007/10/03)
- File number:2
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- 848031-94-7
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Benign-by-design preparation of humin-based iron oxide catalytic nanocomposites
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Green Chemistry p. 4423 - 4434
(2017/09/27)
- File number:6
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- 84804-69-3
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INHIBITORS OF HEPATITIS C VIRUS RNA-DEPENDENT RNA POLYMERASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME
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- File number:2
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- 84807-09-0
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Synthesis of C4-Aminated Indoles via a Catellani and Retro-Diels-Alder Strategy
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Journal of the American Chemical Society p. 9731 - 9738
(2019/06/24)
- File number:11
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- 84807-10-3
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N4-Unsubstituted N1-Arylpiperazines as High-Affinity 5-HT1A Receptor Ligands
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Journal of Medicinal Chemistry p. 1942 - 1954
(2007/10/02)
- File number:3
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- 84807-26-1
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Design, Synthesis, and Structure-Activity Relationships of Indoline-Based Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-Like 2 (Keap1-Nrf2) Protein-Protein Interaction Inhibitors
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Journal of Medicinal Chemistry p. 11149 - 11168
(2020/11/09)
- File number:5
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- 848093-05-0
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Evaluation and synthesis of polar aryl- and heteroaryl spiroazetidine-piperidine acetamides as ghrelin inverse agonists
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ACS Medicinal Chemistry Letters p. 156 - 161
(2015/03/04)
- File number:2
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- 848095-02-3
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Base catalyzed reaction of ethyl thioglycolate with β-aryl-β-(methylthio) acroleins: A general method for the synthesis of 2-carbethoxy-5-substituted/4,5-annulated thiophenes in high overall yields
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Tetrahedron Letters p. 928 - 931
(2016/02/05)
- File number:4
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- 848133-75-5
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Irreversible inhibition of epidermal growth factor receptor activity by 3-aminopropanamides
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Journal of Medicinal Chemistry p. 2251 - 2264
(2012/05/20)
- File number:13
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- 848133-87-9
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Optimization of 6,7-disubstituted-4-(arylamino)quinoline-3-carbonitriles as orally active, irreversible inhibitors of human epidermal growth factor receptor-2 kinase activity
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Journal of Medicinal Chemistry p. 1107 - 1131
(2007/10/03)
- File number:4
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- 84814-09-5
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New silicon precursor compounds and method for fabricating silicon-containing thin film using the same
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- File number:2
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- 848141-13-9
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Discovery of a Series of Pyrazinone RORγAntagonists and Identification of the Clinical Candidate BI 730357
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ACS Medicinal Chemistry Letters p. 143 - 154
(2021/01/26)
- File number:10
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- 84814-11-9
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New silicon precursor compounds and method for fabricating silicon-containing thin film using the same
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- File number:2
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- 84815-20-3
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α2 adrenoceptor agonists as potential analgesic agents. 3. Imidazolylmethylthiophenes
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Journal of Medicinal Chemistry p. 863 - 872
(2007/10/03)
- File number:9
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- 848153-29-7
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N-Boc-O-tosyl hydroxylamine as a safe and efficient nitrogen source for the N-amination of aryl and alkyl amines: Electrophylic amination
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Synlett p. 1993 - 1996
(2011/10/08)
- File number:4
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- 848170-22-9
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How do reaction conditions affect the enantiopure synthesis of 2-substituted-1,4-benzodioxane derivatives?
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Chirality p. 943 - 950
(2018/05/16)
- File number:2
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- 848186-83-4
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Synthesis and structure-activity relationships of isoxazole carboxamides as growth hormone secretagogue receptor antagonists
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Bioorganic and Medicinal Chemistry Letters p. 1201 - 1204
(2007/10/03)
- File number:2
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- 848192-92-7
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Benzoxaborole Antimalarial Agents. Part 5. Lead Optimization of Novel Amide Pyrazinyloxy Benzoxaboroles and Identification of a Preclinical Candidate
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Journal of Medicinal Chemistry p. 5889 - 5908
(2017/07/22)
- File number:4
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- 84821-53-4
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SYNTHESIS AND CRYSTAL STRUCTURE OF NONAMETHYLRUTHENOCENYLCARBENIUM HEXAFLUOROPHOSPHATE
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Journal of Organometallic Chemistry p. 229 - 238
(2007/10/02)
- File number:19
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- 848243-23-2
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SULFONAMIDE DERIVATIVES AND USE THEREOF AS VGSC INHIBITORS
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- File number:2
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- 84824-92-0
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Asymmetric synthesis of conformationally constrained cis-1-amino-1-phenylcyclohexan-2-ol
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Tetrahedron Asymmetry p. 1501 - 1506
(2007/10/03)
- File number:3
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- 848258-31-1
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Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor α agonists
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Bioorganic and Medicinal Chemistry Letters p. 4689 - 4693
(2008/02/11)
- File number:8
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- 848259-27-8
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Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor α agonists
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Bioorganic and Medicinal Chemistry Letters p. 4689 - 4693
(2008/02/11)
- File number:8
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- 84828-97-7
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Practical synthesis of (2′ R)-2′-deoxy-2′-C-methyluridine by highly diastereoselective homogeneous hydrogenation
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Journal of Organic Chemistry p. 297 - 300
(2011/03/20)
- File number:47
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- 848316-21-2
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Heteroarylmethoxyphenylalkoxyiminoalkylcarboxylic acids as leukotriene biosynthesis inhibitors
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Journal of Medicinal Chemistry p. 690 - 705
(2007/10/03)
- File number:3
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- 84833-19-2
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Continuous flow photochemistry as an enabling synthetic technology: Synthesis of substituted-6(5: H)-phenanthridinones for use as poly(ADP-ribose) polymerase inhibitors
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MedChemComm p. 720 - 724
(2016/05/19)
- File number:5
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- 848357-95-9
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TETRACYCLIC HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES
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- File number:3
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- 848369-52-8
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A General synthetic procedure for 2-chloromethyl-4(3H)-quinazolinone derivatives and their utilization in the preparation of novel anticancer agents with 4-anilinoquinazoline scaffolds
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Molecules p. 9473 - 9485
(2011/02/27)
- File number:6
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- 848472-44-6
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Sulfonylureido thiazoles as fructose-1,6-bisphosphatase inhibitors for the treatment of Type-2 diabetes
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Bioorganic and Medicinal Chemistry Letters p. 594 - 599
(2010/05/19)
- File number:11
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- 848482-93-9
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Disubstituted pyrimidines as Lck inhibitors
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Bioorganic and Medicinal Chemistry Letters p. 5440 - 5443
(2010/04/26)
- File number:6
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- 848488-74-4
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DIHYDROPYRIMIDINE COMPOUNDS AND THEIR APPLICATION IN PHARMACEUTICALS
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- File number:4
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- 848488-91-5
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Small Molecule Inhibitors of Metabolic Enzymes Repurposed as a New Class of Anthelmintics
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ACS Infectious Diseases p. 1130 - 1145
(2018/05/15)
- File number:6
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- 848499-31-0
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Discovery of potent and liver-targeted stearoyl-CoA desaturase (SCD) inhibitors in a bispyrrolidine series
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Bioorganic and Medicinal Chemistry Letters p. 980 - 984
(2012/03/26)
- File number:7
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- 848501-94-0
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HETEROCYCLYL-SUBSTITUTED ANTI-HYPERCHOLESTEROLEMIC COMPOUNDS
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- File number:8
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- 848579-43-1
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Radical scavenging and antibacterial activity of caffemides against gram positive, gram negative and clinical drug resistance bacteria
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Bioorganic and Medicinal Chemistry Letters p. 5943 - 5946
(2016/12/06)
- File number:2
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- 84858-98-0
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Ring chain transformations; X: Synthesis of condensed (ω-aminoalkyl)imidazoles by ring chain transformation
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Synthesis p. 521 - 524
(2007/10/02)
- File number:2
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- 848591-89-9
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Octahydropyrrolo[3,4-c]pyrrole: A diamine scaffold for construction of either α4β2 or α7-selective nicotinic acetylcholine receptor (nAChR) ligands. Substitutions that switch subtype selectivity
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Journal of Medicinal Chemistry p. 4126 - 4141
(2010/03/02)
- File number:4
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- 848642-13-7
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Preparation of α and β anomers of 1,2,3,6-tetra-O-acetyl-4- chloro-4-deoxy-D-galactopyranose based upon anomerization and kinetic acetylation
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Carbohydrate Research p. 489 - 495
(2007/10/03)
- File number:2
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- 84867-81-2
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Regio- and chemoselective conjugate 1,4-reduction of α-oxoketene dithioacetals with sodium borohydride and sodium cyanoborohydride
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Tetrahedron p. 2195 - 2204
(2007/10/02)
- File number:2
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- 848691-22-5
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Discovery of ANA975: An oral prodrug of the TLR-7 agonist isatoribine
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Nucleosides, nucleotides and nucleic acids p. 635 - 640
(2008/09/16)
- File number:5
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- 848694-10-0
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Synthesis and characterization of metabolites and potential impurities of the antiulcerative drug tenatoprazole
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Synthetic Communications p. 1725 - 1736
(2008/09/20)
- File number:3
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- 84871-12-5
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New phenylcyclohexyl- and cyclohexylphenylamines. Synthesis and pharmacological activity
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Farmaco, Edizione Scientifica p. 191 - 202
(2007/10/02)
- File number:2
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- 84877-44-1
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Substituent effects. XX. Highly electron-deficient carbocation solvolyses
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Bulletin of the Chemical Society of Japan p. 1138 - 1145
(2007/10/02)
- File number:4
-